One-Pot Synthesis of Novel 2,3-Dihydro-1H-indazoles

Molecules

关键词: 2,3-dihydro-1H-indazole;    synthesis;    heterocycle;    indazoles;    copper coupling;   

DOI  :  10.3390/molecules16119553

来源: DOAJ

【 摘 要 】

A copper(I)-mediated one-pot synthesis of 2,3-dihydro-1H-indazole heterocycles has been developed. This synthetic route provides the desired indazoles in moderate to good yields (55%–72%) which are substantially better than those achievable with an alternative two-step reaction sequence. The reaction is tolerant of functionality on the aromatic ring.

【 授权许可】

Unknown