Recent advances in the preparation of aziridines and their application in organic synthesis

Química Nova

Sá, Marcus Mandolesi¹  Universidade Federal de Santa Catarina, Florianópolis, Brasil¹  Bisol, Tula Beck¹ 

关键词: aziridines;    synthetic methods;    heterocycles.;   

DOI  :  10.1590/S0100-40422007000100022

学科分类：化学（综合）

来源: Sociedade Brasileira de Quimica

【 摘 要 】

This article surveys a selection of the most recent advances in aziridine synthesis. Novel synthetic methods and new insights into existing methodologies for the selective construction of the title compounds reported in the past decade are discussed in terms of synthetic applicability and environmentally benign conditions. Mechanisms involving stereoselective preparation of structurally diverse aziridines are also presented in order to highlight the most important issues associated with the synthesis of these versatile building blocks.

【 授权许可】

Unknown