Recent advances in the preparation of aziridines and their application in organic synthesis

Quimica nova

Sá, Marcus Mandolesi¹  Bisol, Tula Beck¹ 

[1] Universidade Federal de Santa Catarina, Florianópolis, Brasil

关键词: aziridines;    synthetic methods;    heterocycles.;   

DOI  :  10.1590/S0100-40422007000100022

学科分类：化学（综合）

来源: Sociedade Brasileira de Quimica

【 摘 要 】

This article surveysa selection of the most recent advances in aziridine synthesis. Novel syntheticmethods and new insights into existing methodologies for the selective constructionof the title compounds reported in the past decade are discussed in terms ofsynthetic applicability and environmentally benign conditions. Mechanisms involvingstereoselective preparation of structurally diverse aziridines are also presentedin order to highlight the most important issues associated with the synthesisof these versatile building blocks.

【 授权许可】

CC BY