Synthesis of N-Azaaryl Anilines: An Efficient Protocol via Smiles Rearrangement

Bulletin of the Korean chemical society

Dong-Soo Shin¹  Hua Zuo¹  Xiao-Yan He¹  Heng-Zhi Sun¹  Xiu-Hua Wang¹  Ki-Cheol Mun¹  Huan Yue¹  Yin Wang¹  Di Hou¹  B. Prem Kumar¹  Jia-Lian Tan¹  Shuai Xia¹  Li-Ying Wang¹ 

关键词: Smiles rearrangement;    N-Azaaryl anilines;    Amine;    Phenol;    Synthesis;   

DOI  :  

学科分类：化学（综合）

来源: Korean Chemical Society

【 摘 要 】

An efficient process for the synthesis of N-azaaryl anilines via Smiles rearrangement as a tool. A variety of Nazaaryl anilines were generated by the reaction of substituted phenols, substituted anilines, aminopyridines and chloroacetyl chloride or pyridols, under base condition in good to excellent yields.

【 授权许可】

Unknown